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Tapentadol is a prescription medication used to manage moderate to severe pain. It combines two mechanisms of action: it is a mu-opioid receptor agonist and also inhibits the reuptake of norepinephrine. Tapentadol is used to treat moderate to severe pain, including pain from injuries, surgeries, or certain medical conditions. It is often prescribed when other pain relievers are not effective or suitable. It is available in extended-release tablets (for continuous pain relief) and immediate-release tablets (for acute pain).

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